Structure-activity relationships of new aranorosin analogs to antifungal activity.

نویسندگان

  • E K Vijayakumar
  • K Roy
  • S Chatterjee
  • T Mukhopadhyay
  • R G Bhat
  • B N Ganguli
چکیده

prepared by stirring a mixture of 1 with the corresponding carboxylic acid (1.1 equiv.) in the presence of dicyclohexylcarbodiimide (DCC) (1.1 equiv.) and 4-dimethylaminopyridine (DMAP) (0.1 equiv.) in CH2Cl2 at room temperature for 24 hours. The crude products, obtained after usual work up, were purified by preparative TLC on silica gel (Article No. 13794, E. Merck) using CHCl3 MeOH (9:1) as the developing solvent.

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عنوان ژورنال:
  • The Journal of antibiotics

دوره 51 5  شماره 

صفحات  -

تاریخ انتشار 1998